• merck millipore,默克密理博,539522,PKCε Translocation Inhibitor Peptide - Calbiochem
  • merck millipore,默克密理博,539522,PKCε Translocation Inhibitor Peptide - Calbiochem

    产品名称:PKCε Translocation Inhibitor Peptide - Calbiochem
    产品型号:539522
    The PKCε Translocation Inhibitor Peptide, Negative Control controls the biological activity of PKCε. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosp More>>

    merck millipore,默克密理博,539522,PKCε Translocation Inhibitor Peptide - Calbiochem

  • 产品介绍
  • merck millipore,默克密理博,539522,PKCε Translocation Inhibitor Peptide - Calbiochem

    重要规格表

    经验配方
    C₃₇H₆₅N₉O₁₃
    描述
    概述 An octapeptide that selectively inhibits the translocation of protein kinase Cε to subcellular sites in a reversible manner. Inhibition of PKCε translocation is known to specifically block phorbol ester- or norepinephrine-mediated regulation of contraction in cardiomyocytes.
    产品目录编号 539522
    品牌系列 Calbiochem®
    同义词 Protein Kinase Cε Translocation Inhibitor I, EAVSLKPT, PKCε Translocation Inhibitor I, PKCε-RACK2 Interaction Inhibitor I
    参考
    参考 Yedovitzky, M., et al. 1997. J. Biol. Chem. 272, 1417.
    Johnson, J.A., et al. 1996. J. Biol. Chem. 271, 24962.
    产品信息
    具有ATP竞争性 N
    声明 Sold under license of U.S. Patent 5,783,405.
    形式 White lyophilized solid
    配方 Supplied as a trifluoroacetate salt.
    Hill配方 C₃₇H₆₅N₉O₁₃
    化学配方 C₃₇H₆₅N₉O₁₃
    Molar Mass 844.0
    吸湿 Hygroscopic
    肽序列 H-Glu-Ala-Val-Ser-Leu-Lys-Pro-Thr-OH
    可逆 Y
    生物信息
    主靶 PKCε Translocation
    纯度 ≥97% by HPLC
    理化信息
    细胞可渗透 N
    溶解度 H₂O
    肽序列 H-Glu-Ala-Val-Ser-Leu-Lys-Pro-Thr-OH
    储存和货运信息
    货运代码 Ambient Temperature Only
    毒性 Standard Handling
    储存 +2°C to +8°C
    吸湿 Hygroscopic
    无需冷冻 No
    特殊指南 Following reconstitution, aliquot and freeze (-20°C) for long-term storage. Stock solutions are stable for up to 6 months at -20°C.

    merck millipore,默克密理博,539522,PKCε Translocation Inhibitor Peptide - Calbiochem

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