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merck millipore,默克密理博,573129,InSolution™ STAT3 Inhibitor III, WP1066 - Calbiochem
产品名称:InSolution™ STAT3 Inhibitor III, WP1066 - Calbiochem
产品型号:573129
The InSolution™ STAT3 Inhibitor III, WP1066, also referenced under CAS 857064-38-1, controls the biological activity of STAT3. This small molecule/inhibitor is primarily used for Phosphorylation & Dep More>>
merck millipore,默克密理博,573129,InSolution™ STAT3 Inhibitor III, WP1066 - Calbiochem
- 产品介绍
重要规格表
经验配方 C₁₇H₁₄BrN₃O 描述 概述 A cell-permeable AG 490 (Cat. No. 658401) tyrphostin analog that acts as an effective STAT3 pathway inhibitor and a much more potent antitumor agent than AG 490 in inhibiting malignant glioma growth both in cultures in vitro (IC50 = 5.6 and 3.7 µM in a viability assay using U87-MG and U373-MG, respectively; no inhibition against nontumor NHA at 10 µM) and in mice in vivo. Shown to cross blood-brain barrier in mice in vivo. 产品目录编号 573129 品牌系列 Calbiochem®
参考 参考 Iwamaru, A., et al. 2007. Oncogene, 26, 2435. 产品信息 形式 Liquid 配方 A 50 mM (5 mg/281 µl) solution of STAT3 Inhibitor III, WP1066 (Cat. No. 573097) in DMSO. Hill配方 C₁₇H₁₄BrN₃O 化学配方 C₁₇H₁₄BrN₃O Molar Mass 356.2 吸湿 Hygroscopic
结构配方图像 生物信息 纯度 ≥97% by HPLC 安全信息 R相 R: 36/38
Irritating to eyes and skin.储存和货运信息 货运代码 Dry Ice Only
毒性 Irritant
储存 -20°C
避光 Protect from light
吸湿 Hygroscopic
无需冷冻 No
特殊指南 Following intial thaw, aliquot and freeze (-20°C). 包装信息 惰性气体下包装 Packaged under inert gas
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