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merck millipore,默克密理博,506148,InSolution™ p38 MAP Kinase Inhibitor III - Calbiochem
产品名称:InSolution™ p38 MAP Kinase Inhibitor III - Calbiochem
产品型号:506148
The InSolution™ p38 MAP Kinase Inhibitor III controls the biological activity of p38 MAP Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
merck millipore,默克密理博,506148,InSolution™ p38 MAP Kinase Inhibitor III - Calbiochem
- 产品介绍
重要规格表
经验配方 C₂₃H₂₁FN₄S 描述 产品目录编号 506148 品牌系列 Calbiochem®
参考 参考 Laufer, S.A., et al. 2003. J. Med. Chem. 46, 3230. 产品信息 具有ATP竞争性 Y 形式 Liquid 配方 A 10 mM (1 mg/247 µl) solution of p38 MAP Kinase Inhibitor III (Cat. No. 506121) in DMSO. Hill配方 C₂₃H₂₁FN₄S 化学配方 C₂₃H₂₁FN₄S Molar Mass 404.5 吸湿 Hygroscopic
可逆 Y 结构配方图像 生物信息 主靶 p38 MAP kinase 主靶IC50 0.38 µM for p38α; 0.16 and 0.039 µM in suppressing LPS-induced TNF-α and IL-1β release, respectively, in human PBMC; ED50 = 1.33 mg/kg in suppressing LPS-induced TNF-α release in mouse 纯度 ≥98% by HPLC 理化信息 细胞可渗透 Y 储存和货运信息 货运代码 Shipped with Blue Ice or with Dry Ice
毒性 Standard Handling
储存 +2°C to +8°C
避光 Protect from light
吸湿 Hygroscopic
无需冷冻 No
特殊指南 Following initial use, aliquot and refrigerate (4°C). 包装信息 惰性气体下包装 Packaged under inert gas
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