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merck millipore,默克密理博,371725,GPR43 (FFA2) Agonist - Calbiochem
产品名称:GPR43 (FFA2) Agonist - Calbiochem
产品型号:371725
The GPR43 (FFA2) Agonist controls the biological activity of GPR43. This small molecule/inhibitor is primarily used for Biochemicals applications.
merck millipore,默克密理博,371725,GPR43 (FFA2) Agonist - Calbiochem
- 产品介绍
重要规格表
经验配方 C₂₁H₂₁ClN₂OS 描述 概述 A phenylacetamide compound that acts as an allosteric agonist of FFA2 (GPR43), demonstrating a left-shifted acetate dose response (IC50 = 0.7 µM) and 111% efficacy relative to acetate in hFFA2 forskolin-induced cAMP assays. 产品目录编号 371725 品牌系列 Calbiochem®
同义词 (S)-2-(4-chlorophenyl)-3,3-dimethyl-N-(5-phenylthiazol-2-yl)butanamide 参考 参考 Wang, Y., et al. 2009. Bioorg. Med. Chem. Lett. 20, 493. 产品信息 形式 White solid Hill配方 C₂₁H₂₁ClN₂OS 化学配方 C₂₁H₂₁ClN₂OS Molar Mass 384.92 结构配方图像 生物信息 纯度 >95% by HPLC 理化信息 溶解度 DMSO 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Regulatory Review
储存 +2°C to +8°C
无需冷冻 No
特殊指南 Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
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