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经验配方 CAS号 C₁₄H₁₂BrN₅ 171179-06-9 描述 产品目录编号 513036 品牌系列 Calbiochem®
参考 参考 Cunnick, J.M., et al. 1998. J. Biol. Chem. 273, 14468.
Rewcastle, G.W., et al. 1998. J. Med. Chem. 41, 742.产品信息 CAS号 171179-06-9 具有ATP竞争性 Y 形式 Liquid 配方 A 10 mM (500 µg/151 µl) solution of PD 158780 (Cat. No. 513035) in DMSO. Hill配方 C₁₄H₁₂BrN₅ 化学配方 C₁₄H₁₂BrN₅ Molar Mass 330.2 吸湿 Hygroscopic
可逆 Y 结构配方图像 生物信息 主靶 EGFR 主靶IC50 8 pM against EGFR tyrosine kinase activity; 49 nM, 52 nM, against heregulin-stimulated autophosphorylation in SK-BR-3 and MDA-MB-453 breast carcinomas, respectively 纯度 ≥95% by HPLC 理化信息 细胞可渗透 Y 储存和货运信息 货运代码 Shipped with Blue Ice or with Dry Ice
毒性 Standard Handling
储存 -20°C
避光 Protect from light
吸湿 Hygroscopic
无需冷冻 No
特殊指南 Following initial thaw, aliquot and freeze (-20°C). 包装信息 惰性气体下包装 Packaged under inert gas
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