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merck millipore,默克密理博,219457,Cdk Inhibitor, p35 - CAS 471270-60-7 - Calbiochem
产品名称:Cdk Inhibitor, p35 - CAS 471270-60-7 - Calbiochem
产品型号:219457
The Cdk Inhibitor, p35, also referenced under CAS 471270-60-7, controls the biological activity of Cdk. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applicat More>>
merck millipore,默克密理博,219457,Cdk Inhibitor, p35 - CAS 471270-60-7 - Calbiochem
- 产品介绍
重要规格表
经验配方 CAS号 C₁₈H₂₄N₆O₂ 471270-60-7 描述 概述 An analog of Olomoucine (Cat. No. 495620) that acts as a potent inhibitor of Cdk1 (IC50 = 100 nM) and Cdk2 (IC50 = 80 nM). Also displays anti-proliferative and pro-apoptotic effects. The correlation between inhibition of Cdk1/Cdk2 and inhibition of cell proliferation suggests that the anti-proliferative effects are due, in part, to Cdk inhibition. 产品目录编号 219457 品牌系列 Calbiochem®
同义词 2-(3-Hydroxypropylamino)-6-(o-hydroxybenzylamino)-9-isopropylpurine 参考 参考 Vermeulen, K., et al. 2002. Leukemia 16, 299. 产品信息 CAS号 471270-60-7 具有ATP竞争性 N 形式 Yellow solid Hill配方 C₁₈H₂₄N₆O₂ 化学配方 C₁₈H₂₄N₆O₂ Molar Mass 356.4 可逆 N 结构配方图像 生物信息 主靶 CDK1, CDK2 主靶IC50 100 nM, 80 nM, against Cdk1 and Cdk2, respectively 纯度 ≥95% by HPLC 理化信息 细胞可渗透 N 溶解度 DMSO 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Standard Handling
储存 -20°C
避光 Protect from light
无需冷冻 No
特殊指南 Following reconstitution aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C. 包装信息 惰性气体下包装 Packaged under inert gas
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