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merck millipore,默克密理博,513020,PD 145065 - CAS 153049-49-1 - Calbiochem
产品名称：PD 145065 - CAS 153049-49-1 - Calbiochem
产品型号：513020
A highly potent but non-selective endothelin receptor antagonist [IC₅₀= 4 nM for the ETA receptor (rabbit renal artery vascular smooth muscle cells); IC₅₀ = 15 nM for the ETB receptor (rat More>>
merck millipore,默克密理博,513020,PD 145065 - CAS 153049-49-1 - Calbiochem
- 产品介绍
重要规格表
经验配方 CAS号 C₅₂H₆₃N₇O₁₀ · 2Na 153049-49-1 描述 概述 A highly potent but non-selective endothelin receptor antagonist [IC50 = 4 nM for the ETA receptor (rabbit renal artery vascular smooth muscle cells); IC50 = 15 nM for the ETB receptor (rat cerebellum)]. 产品目录编号 513020 品牌系列 Calbiochem®
参考 参考 Han, H.K., et al. 1998. Life Sci. 63, 1599.
Allcock, G.H., et al. 1995. Br. J. Pharmacol. 116, 2482.
Wellings, R.P., et al. 1994. Eur. J. Pharmacol. 256, 201.
Cody, W.L., et al. 1993. Med. Chem. Res. 3, 154.
Doherty, A.M., et al. 1993. J. Cardiovasc. Pharmacol. 22, S98 (Suppl.).产品信息 CAS号 153049-49-1 具有ATP竞争性 N 形式 White solid Hill配方 C₅₂H₆₃N₇O₁₀ · 2Na 化学配方 C₅₂H₆₃N₇O₁₀ · 2Na Molar Mass 992.1 肽序列 Ac-D-Bhg-Leu-Asp-Ile-Ile-Trp-OH (Bhg = 5H-dibenzo[a,d]cycloheptene-5-glycine) 可逆 N 生物信息 主靶 Endothelin receptor antagonist 主靶IC50 4 nM against endothelin receptor (ETA receptor) in rabbit renal artery vascular smooth muscle cells; 15 nM for the ETB receptor (rat cerebellum) 纯度 ≥98% by HPLC 理化信息 细胞可渗透 N 溶解度 Phosphate Buffer, pH 7.5 肽序列 Ac-D-Bhg-Leu-Asp-Ile-Ile-Trp-OH (Bhg = 5H-dibenzo[a,d]cycloheptene-5-glycine) 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Standard Handling
储存 +2°C to +8°C
无需冷冻 No
特殊指南 Following reconstitution, aliquot and freeze (-20°C) for long-term storage. Stock solutions are stable for up to 4 months at -20°C. Avoid freeze/thaw cycles of solutions.
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