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经验配方 CAS号 C₆₇H₁₂₄N₁₈O₁₅ 145854-59-7 描述 概述 A cell-permeable, amphiphilic, mastoparan analog with five-fold greater potency than Mastoparan Cat. No. 444898. An activator of α-subunit of G-proteins. Evokes rapid upregulation of FAK tyrosine phosphorylation via activation of G-proteins. 产品目录编号 444896 品牌系列 Calbiochem®
参考 参考 Mironov, S.L., and Richter, D.W. 2000. Brain Res. 853, 60.
Park, H.S., et al. 2000. Biochim. Biophys. Acta 1484, 151.
Zhang, C., et al. 1996. FEBS Lett. 386, 185.
Leyte, A., et al. 1992. EMBO J. 11 4795.
Higashijima, T., et al. 1990. J. Biol. Chem. 265, 14176.产品信息 CAS号 145854-59-7 具有ATP竞争性 N 形式 White solid 配方 Supplied as a trifluoroacetate salt. Hill配方 C₆₇H₁₂₄N₁₈O₁₅ 化学配方 C₆₇H₁₂₄N₁₈O₁₅ Molar Mass 1421.8 肽序列 H-Ile-Asn-Leu-Lys-Ala-Leu-Ala-Ala-Leu-Ala-Lys-Ala-Leu-Leu-NH₂ 可逆 N 基于肽含量售出 Yes
生物信息 主靶 α-subunit of G-proteins 纯度 ≥98% by HPLC 理化信息 细胞可渗透 Y 溶解度 H₂O 肽含量 Yes
肽序列 H-Ile-Asn-Leu-Lys-Ala-Leu-Ala-Ala-Leu-Ala-Lys-Ala-Leu-Leu-NH₂ 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Standard Handling
储存 -20°C
无需冷冻 No
特殊指南 Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
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