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经验配方 CAS号 C₁₁H₈N₂ 161468-32-2 描述 概述 A potent, cell-permeable, reversible, and specific inhibitor of protein kinase A (IC50 = 30 nM). Inhibition is competitive with respect to ATP. Shows only weak inhibitory activities against Ca2+-dependent protein kinase (CDPK), MLCK, PKC, and cyclic nucleotide-binding phosphatase. 产品目录编号 238900 品牌系列 Calbiochem®
同义词 PKA Inhibitor XI 参考 参考 Lu, Z.X., et al. 1996. Biol. Chem. Hoppe Seyler 377, 373. 产品信息 CAS号 161468-32-2 具有ATP竞争性 Y 形式 White solid Hill配方 C₁₁H₈N₂ 化学配方 C₁₁H₈N₂ Molar Mass 168.2 可逆 Y 结构配方图像 生物信息 主靶 PKA 主靶IC50 30 nM against protein kinase A 纯度 ≥95% by HPLC 理化信息 细胞可渗透 Y 溶解度 DMSO 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Standard Handling
储存 +2°C to +8°C
无需冷冻 No
特殊指南 Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C. 包装信息 惰性气体下包装 Packaged under inert gas
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