- 当前位置:首页 > >Merck Millipore > 生命科学研究
- 生命科学研究
-

-
merck millipore,默克密理博,218710,Casein Kinase II Inhibitor III, TBCA - CAS 934358-00-6 - Calbiochem
产品名称:Casein Kinase II Inhibitor III, TBCA - CAS 934358-00-6 - Calbiochem
产品型号:218710
The Casein Kinase II Inhibitor III, TBCA, also referenced under CAS 934358-00-6, controls the biological activity of Casein Kinase II. This small molecule/inhibitor is primarily used for Phosphorylati More>>
merck millipore,默克密理博,218710,Casein Kinase II Inhibitor III, TBCA - CAS 934358-00-6 - Calbiochem
- 产品介绍
重要规格表
经验配方 CAS号 C₉H₄Br₄O₂ 934358-00-6 描述 概述 A cell-permeable tetrabrominated cinnamic acid compound that acts as a potent and ATP-competitive inhibitor of Casein Kinase II (IC50 = 110 nM, Ki = 77 nM) with greater selectivity than TBB (Cat. Nos. 218697 and 218708) and DMAT (Cat. Nos. 218699 and 218706) against a panel of 28 commonly studied kinases. Shown to efficiently induces apoptosis in Jurkat cells (DC50 = 7.7 µM). Also available as a 25 mM solution in DMSO (Cat. No. 218861). 产品目录编号 218710 品牌系列 Calbiochem®
同义词 (E)-3-(2,3,4,5-Tetrabromophenyl)acrylic acid, CKII Inhibitor, TBCA 参考 参考 Pagano, M.A., et al. 2006. Chembiochem 8, 129 产品信息 CAS号 934358-00-6 具有ATP竞争性 Y 形式 Off-white solid Hill配方 C₉H₄Br₄O₂ 化学配方 C₉H₄Br₄O₂ Molar Mass 463.8 可逆 N 结构配方图像 生物信息 主靶 Casein Kinase II 主靶IC50 110 nM 主靶Ki 77 nM against Casein Kinase II 纯度 ≥95% by HPLC 理化信息 细胞可渗透 Y 溶解度 DMSO or EtOH 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Irritant
储存 +2°C to +8°C
避光 Protect from light
无需冷冻 No
特殊指南 Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C. 包装信息 惰性气体下包装 Packaged under inert gas
上一件merck millipore产品:merck millipore,默克密理博,AB3081,Anti-Na+/H+ Exchanger-1 Antibody
下一件merck millipore产品:merck millipore,默克密理博,437629,Lipopolysaccharide, Salmonella minnesota Re 595 - Calbiochem
merck millipore,默克密理博,524748,PDE4D Inhibitor, GEBR-7b - Calbiochem
merck millipore,默克密理博,05-1149,Anti-ADP-Ribosylation Factor 6 Antibody, clone 6ARF01
merck millipore,默克密理博,416154,Pre-mRNA Splicing Inhibitor, Isoginkgetin - CAS 548-19-6 - Calbiochem
merck millipore,默克密理博,100107,A23187, 4-Bromo- - CAS 76455-82-8 - Calbiochem
merck millipore,默克密理博,AB3081,Anti-Na+/H+ Exchanger-1 Antibody
merck millipore,默克密理博,437629,Lipopolysaccharide, Salmonella minnesota Re 595 - Calbiochem
merck millipore,默克密理博,04-1035,Anti-SMAD3 Antibody, clone EP568Y, rabbit monoclonal
merck millipore,默克密理博,MAB3310,Anti-TIMP-2 Antibody, clone 67-4H11
merck millipore,默克密理博,MSBVN1250,MultiScreenHTS BV,1.2 µm,无色,非无菌
merck millipore,默克密理博,527460,PhosphoDetect™ Anti-PKR (pThr⁴⁵¹) Rabbit pAb


