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经验配方 K₂[VO(O₂)₂C₆H₄NO₃] · 4H₂O 描述 概述 A potent phosphotyrosine phosphatase inhibitor. Activates the insulin receptor kinase (IRK) of hepatoma cells. Also stimulates lipogenesis in isolated adipocytes. Also reported to potently inhibit PTEN (IC50 = 14 nM). 产品目录编号 203701 品牌系列 Calbiochem®
同义词 Dipotassium Bisperoxo(5-hydroxypyridine-2-carboxyl)oxovanadate (V), PTEN Inhibitor III, PTP Inhibitor XV 参考 参考 Schmid, A.C., et al. 2004. FEBS Lett. 566, 35.
Posner, B.I., et al. 1994. J. Biol. Chem. 269, 4596.产品信息 具有ATP竞争性 N 形式 Yellow solid Hill配方 K₂[VO(O₂)₂C₆H₄NO₃] · 4H₂O 化学配方 K₂[VO(O₂)₂C₆H₄NO₃] · 4H₂O Molar Mass 419.3 可逆 N 结构配方图像 生物信息 主靶 PTEN 主靶IC50 14 nM 纯度 ≥70% by ⁵¹V-NMR 理化信息 细胞可渗透 N 溶解度 H₂O 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Standard Handling
储存 -20°C
避光 Protect from light
无需冷冻 No
特殊指南 Unstable in solution; reconstitute just prior to use. 包装信息 惰性气体下包装 Packaged under inert gas
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