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merck millipore,默克密理博,182540,Aromatase Inhibitor I - CAS 331684-05-0 - Calbiochem
产品名称:Aromatase Inhibitor I - CAS 331684-05-0 - Calbiochem
产品型号:182540
The Aromatase Inhibitor I, also referenced under CAS 331684-05-0, controls the biological activity of Aromatase.
merck millipore,默克密理博,182540,Aromatase Inhibitor I - CAS 331684-05-0 - Calbiochem
- 产品介绍
重要规格表
经验配方 CAS号 C₁₇H₁₁N₃O₄ 331684-05-0 描述 概述 A potent, competitive, nonsteroidal inhibitor of aromatase (P450arom; IC50 = 40 nM for human aromatase). Reported to be more potent than fadrozole in inhibiting aromatase activity. Does not significantly inhibit 17α-hydroxylase. 产品目录编号 182540 品牌系列 Calbiochem®
同义词 4-(Imidazolylmethyl)-1-nitro-9H-9-xanthenone 参考 参考 Recanatini, M., et al. 2001. J. Med. Chem. 44, 672. 产品信息 CAS号 331684-05-0 具有ATP竞争性 Y 形式 White solid Hill配方 C₁₇H₁₁N₃O₄ 化学配方 C₁₇H₁₁N₃O₄ Molar Mass 321.3 可逆 N 结构配方图像 生物信息 主靶 P450 arom. 主靶IC50 40 nM against P450arom 纯度 ≥95% by HPLC 理化信息 细胞可渗透 N 溶解度 DMSO 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Standard Handling
储存 -20°C
避光 Protect from light
无需冷冻 No
特殊指南 Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C. 包装信息 惰性气体下包装 Packaged under inert gas
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