• merck millipore,默克密理博,565625,SC-68376 - CAS 318480-82-9 - Calbiochem
  • merck millipore,默克密理博,565625,SC-68376 - CAS 318480-82-9 - Calbiochem

    产品名称:SC-68376 - CAS 318480-82-9 - Calbiochem
    产品型号:565625
    A potent, reversible, cell-permeable, ATP-competitive, and selective inhibitor of p38 MAP kinase activity in a dose-dependent manner (IC₅₀ = 2-5 µM).

    merck millipore,默克密理博,565625,SC-68376 - CAS 318480-82-9 - Calbiochem

  • 产品介绍
  • merck millipore,默克密理博,565625,SC-68376 - CAS 318480-82-9 - Calbiochem

    重要规格表

    经验配方 CAS号
    C₁₅H₁₂N₂O318480-82-9
    描述
    概述 A potent, reversible, cell-permeable, ATP-competitive, and selective inhibitor of p38 MAP kinase activity in a dose-dependent manner (IC50 = 2-5 µM). Does not inhibit basal ERK or IL-1-induced JNK activity.
    产品目录编号 565625
    品牌系列 Calbiochem®
    同义词 2-Methyl-4-phenyl-5-(4-pyridyl)oxazole
    参考
    参考 Guan, Z., et al. 1998. J. Biol. Chem. 273, 12901.
    Guan, Z., et al. 1997. J. Biol. Chem. 272, 8083.
    产品信息
    CAS号 318480-82-9
    具有ATP竞争性 Y
    形式 White to yellow semi-solid
    Hill配方 C₁₅H₁₂N₂O
    化学配方 C₁₅H₁₂N₂O
    Molar Mass 236.3
    可逆 Y
    结构配方图像
    生物信息
    主靶 p38MAPK
    主靶IC50 2-5 µM against p38MAP kinase activity
    纯度 ≥98% by HPLC
    理化信息
    细胞可渗透 Y
    溶解度 DMSO
    储存和货运信息
    货运代码 Ambient Temperature Only
    毒性 Standard Handling
    储存 +2°C to +8°C
    无需冷冻 No
    特殊指南 Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 1 month at -20°C.

    merck millipore,默克密理博,565625,SC-68376 - CAS 318480-82-9 - Calbiochem

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