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merck millipore,默克密理博,480402,NFAT Inhibitor - Calbiochem
产品名称:NFAT Inhibitor - Calbiochem
产品型号:480402
The NFAT Inhibitor controls the biological activity of NFAT. This small molecule/inhibitor is primarily used for Inflammation/Immunology applications.
merck millipore,默克密理博,480402,NFAT Inhibitor - Calbiochem
- 产品介绍
重要规格表
经验配方 C₇₅H₁₁₈N₂₀O₂₂S 描述 概述 A highly selective NFAT (Nuclear Factor of Activated T-cells) inhibitor that interferes with calcineurin-NFAT interaction without affecting calcineurin (Cat. No. 539568) phosphatase activity. Inhibits NFAT activation and NFAT-dependent expression of endogenous cytokine genes in T cells, without affecting the expression of other cytokines that require calcineurin but not NFAT. 产品目录编号 480402 品牌系列 Calbiochem®
同义词 MAGPHPVIVITGPHEE 参考 参考 Noguchi, H., et al. 2004. Nat. Med. 10, 305.
Kiani, A., et al. 2001. Blood 98, 1480.
Aramburu, J., et al. 1999. Science 285, 2129.产品信息 具有ATP竞争性 N 形式 Lyophilized solid 配方 Supplied as a trifluoroacetate salt. Hill配方 C₇₅H₁₁₈N₂₀O₂₂S 化学配方 C₇₅H₁₁₈N₂₀O₂₂S Molar Mass 1683.9 吸湿 Hygroscopic
肽序列 H-Met-Ala-Gly-Pro-His-Pro-Val-Ile-Val-Ile-Thr-Gly-Pro-His-Glu-Glu-OH 可逆 N 生物信息 主靶 NFAT (Nuclear Factor of Activated T-cells) 纯度 ≥95% by HPLC 理化信息 细胞可渗透 N 溶解度 H₂O 肽序列 H-Met-Ala-Gly-Pro-His-Pro-Val-Ile-Val-Ile-Thr-Gly-Pro-His-Glu-Glu-OH 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Standard Handling
储存 -20°C
吸湿 Hygroscopic
无需冷冻 No
特殊指南 Following initial thaw, aliquot and freeze (-20°C). Avoid freeze/thaw cycles of solutions. 包装信息 惰性气体下包装 Packaged under inert gas
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