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merck millipore,默克密理博,218728,Caspase-9 Inhibitor III - CAS 403848-57-7 - Calbiochem
产品名称:Caspase-9 Inhibitor III - CAS 403848-57-7 - Calbiochem
产品型号:218728
The Caspase-9 Inhibitor III, also referenced under CAS 403848-57-7, controls the biological activity of Caspase-9. This small molecule/inhibitor is primarily used for Cancer applications.
merck millipore,默克密理博,218728,Caspase-9 Inhibitor III - CAS 403848-57-7 - Calbiochem
- 产品介绍
重要规格表
经验配方 CAS号 C₂₄H₃₅ClN₆O₉ 403848-57-7 描述 概述 A potent, irreversible inhibitor of caspase-9. Reported to reduce myocardial infarct size during reperfusion (~70 nM). 产品目录编号 218728 品牌系列 Calbiochem®
同义词 Ac-LEHD-CMK 参考 参考 Mocanu, M.M., et al. 2000. Br. J. Pharmacol. 130, 197. 产品信息 CAS号 403848-57-7 具有ATP竞争性 N 形式 White solid 配方 Supplied as a trifluoroacetate salt. Hill配方 C₂₄H₃₅ClN₆O₉ 化学配方 C₂₄H₃₅ClN₆O₉ Molar Mass 587.0 肽序列 Ac-Leu-Glu-His-Asp-CMK 可逆 N 结构配方图像 生物信息 主靶 caspase-9 主靶IC50 70 nM against caspase-9 纯度 ≥95% by HPLC 理化信息 细胞可渗透 Y 溶解度 DMSO or H₂O 肽序列 Ac-Leu-Glu-His-Asp-CMK 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Standard Handling
储存 -20°C
防潮 Protect from moisture
无需冷冻 No
特殊指南 Following reconstitution aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
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