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merck millipore,默克密理博,368055,Granzyme B Inhibitor II - CAS 1258003-96-1 - Calbiochem
产品名称:Granzyme B Inhibitor II - CAS 1258003-96-1 - Calbiochem
产品型号:368055
The Granzyme B Inhibitor II, also referenced under CAS 1258003-96-1, controls the biological activity of Granzyme B. This small molecule/inhibitor is primarily used for Cancer applications.
merck millipore,默克密理博,368055,Granzyme B Inhibitor II - CAS 1258003-96-1 - Calbiochem
- 产品介绍
重要规格表
经验配方 CAS号 C₂₁H₃₄N₄O₁₀ 1258003-96-1 描述 概述 A potent, reversible inhibitor of granzyme B and caspase-8 (Ki = 1 nM). Also inhibits caspase-1 (<6 nM), caspase-6 (5.6 nM), and caspase-10 (27 nM). 产品目录编号 368055 品牌系列 Calbiochem®
同义词 Caspase-8 Inhibitor I, Ac-IETD-CHO 参考 参考 Gao, C.F., et al. 2001. Exp. Cell. Res. 265, 145.
Garcia-Calvo, M., et al. 1998. J. Biol. Chem. 273, 32608.
Han, Z., et al. 1997. J. Biol. Chem. 272, 13422.产品信息 CAS号 1258003-96-1 具有ATP竞争性 N 形式 White lyophilized solid Hill配方 C₂₁H₃₄N₄O₁₀ 化学配方 C₂₁H₃₄N₄O₁₀ Molar Mass 502.5 肽序列 Ac-Ile-Glu-Thr-Asp-CHO 可逆 Y 结构配方图像 生物信息 主靶 caspase-8 主靶Ki 1 nM against caspase-8 纯度 ≥95% by HPLC 理化信息 细胞可渗透 N 溶解度 DMSO 肽序列 Ac-Ile-Glu-Thr-Asp-CHO 储存和货运信息 货运代码 Ambient Temperature Only
毒性 Standard Handling
储存 -20°C
无需冷冻 No
特殊指南 Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
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