merck millipore,默克密理愽
  • merck millipore,默克密理博,119152,Adenosine A₃ Receptor Antagonist, MRS 1523 - CAS 212329-37-8 - Calbiochem

  • merck millipore,默克密理博,119152,Adenosine A₃ Receptor Antagonist, MRS 1523 - CAS 212329-37-8 - Calbiochem

    产品名称：Adenosine A₃ Receptor Antagonist, MRS 1523 - CAS 212329-37-8 - Calbiochem
    产品型号：119152


    merck millipore,默克密理博,119152,Adenosine A₃ Receptor Antagonist, MRS 1523 - CAS 212329-37-8 - Calbiochem

  • 产品介绍
  • merck millipore,默克密理博,119152,Adenosine A₃ Receptor Antagonist, MRS 1523 - CAS 212329-37-8 - Calbiochem

    重要规格表

    经验配方 CAS号
    C₂₃H₂₉NO₃S 212329-37-8
    描述
    概述 A pyridine derivative that acts as a highly selective antagonist of A3 receptor with excellent potency in both humans and rodents (Ki = 18.9 nM for human A3R, and 113 nM for rat A3R). Exhibits only a trivial antagonistic activity towards A1 and A2A receptors (Ki = 15.6 µM and 2.05 µM for rat A1R and A2AR, respectively). Abolishes the agonistic effects of Cl-IB-MECA (Cat. No. 119139) on A3R-mediated proliferation of primary human coronary smooth muscle cells. Also, reported to block NECA (Cat. No. 119140)-induced bronchoconstriction in an allergic murine model.
    产品目录编号 119152
    品牌系列 Calbiochem®
    同义词 3-propyl-6-ethyl-5[(ethylthio)carbonyl]-2-phenyl-4-propyl-3-pyridine-carboxylate, MRS 1523, MRS-1523
    参考
    参考 Chen, Z., 2012. FASEB J. 26, 1855.
    Chanyshev, B., et al. 2012. Pharmacol Res.65, 338.
    Choi, I., et al. 2011. Am J Pathol. 179, 2042.
    Fan, M., et al. 2003. Am J Physiol Lung Cell Mol Physiol. 284, L1012.
    Li, A. H., et al. 1998. J Med Chem. 41, 3186.
    Jacobson, K. A., et al. 1999. Drug Dev Res. 45, 113.
    产品信息
    CAS号 212329-37-8
    形式 Clear, colorelss oil
    Hill配方 C₂₃H₂₉NO₃S
    化学配方 C₂₃H₂₉NO₃S
    Molar Mass 399.55
    可逆 Y
    结构配方图像
    生物信息
    主靶 A₃ Receptor
    主靶Ki 18.9 nM
    纯度 ≥95% by HPLC
    理化信息
    溶解度 DMSO
    储存和货运信息
    货运代码 Shipped at Ambient Temperature or with Blue Ice or with Dry Ice
    毒性 Standard Handling
    储存 +2°C to +8°C
    避光 Protect from light
    无需冷冻 No
    特殊指南 Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
    包装信息
    惰性气体下包装 Packaged under inert gas

    merck millipore,默克密理博,119152,Adenosine A₃ Receptor Antagonist, MRS 1523 - CAS 212329-37-8 - Calbiochem

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下一件merck millipore产品：merck millipore,默克密理博,AB5458,Anti-Neprilysin Antibody (Neutral Endopeptidase, Nep)


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